Ring-opening and cyclization of aziridines with aryl azides: metal-free synthesis of 6-(triflyloxy)quinolines

文献情報

出版日 2018-10-25

DOI 10.1039/C8QO00984H

インパクトファクター 5.281

著者

Xincheng Li, Boshun Wan

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要旨

Ring-opening and cyclization of aziridines with aryl azides in the presence of TfOH has been developed. This strategy enables the construction of 6-(triflyloxy)quinoline cores by utilizing aziridine as a two-carbon surrogate. The introduction of a trifyl group at the 6-position of quinoline would allow further construction of carbon–carbon and carbon–heteroatom bonds in the cross-coupling reactions.

掲載誌

Organic Chemistry Frontiers

CiteScore: 7.8

自己引用率: 8.7%

年間論文数: 724

Organic Chemistry Frontiers publishes high-quality research from across organic chemistry. Emphases are placed on studies that make significant contributions to the field of organic chemistry by reporting either new or significantly improved protocols or methodologies. Topics include, but are not limited to the following: Organic synthesis Development of synthetic methodologies Catalysis Natural products Functional organic materials Supramolecular and macromolecular chemistry Physical and computational organic chemistry

Ring-opening and cyclization of aziridines with aryl azides: metal-free synthesis of 6-(triflyloxy)quinolines

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